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publicationDate 2008-08-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2008534074-A
titleOfInvention Composition and method of administering rapamycin analogs using medical devices for long-term efficacy
abstract Disclosed are systems and compositions comprising zotarolimus that are safe, effective, and less prone to inflammation compared to the rapamycin and paclitaxel systems. A medical device having a support structure comprising or capable of supporting a pharmaceutically acceptable carrier or excipient, wherein the carrier or excipient may comprise one or more therapeutic agents or substances, the carrier comprising a surface There is a coating on top, which has a therapeutic compound such as a pharmaceutical. Support structures for medical devices include coronary stents, peripheral stents, catheters, arteriovenous grafts, bypass grafts and drug delivery balloons used in the vascular system. These compositions and systems include antiproliferative agents, antiplatelet agents, anti-inflammatory agents, antithrombotic agents, cytotoxic agents, agents that inhibit cytokines or chemokine binding, cell dedifferentiation inhibitors, antihyperlipidemic agents, matrices It can be used in combination with other drugs such as metalloprotease inhibitors, cytostatics or combinations of these and other drugs.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419583338
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507591
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396424
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF6RKC1
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID738078
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20344
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426079355
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ99372
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480166
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410862584
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415732204
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3108
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6918289
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5280961
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD3ZQL7
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25639
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22777
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID607661
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2280
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5311101
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP54320
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419494344
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5I6E3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A3Q1MBI9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13909
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413998864
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID97226
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XT80
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24617
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100038778
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410135424
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25619
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403985
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1401
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419588071
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID104762
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395837
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID744785
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492800
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451708054
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5554
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3672
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1983
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP02776
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A452DIJ9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13726
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492855
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5555
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID91450784
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57352570
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396842
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID104799
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431610529
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22775
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16109
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5743
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492594
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11506004
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO94811
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44259
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3899
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3569
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502717
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451961693
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426080486
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152743203
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25651
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP14847
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26893
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5354357
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22419
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419584599
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5281078
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16581
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP79341
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID14225
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID14068
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71300397
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06579
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP98106
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395337
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41693
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18787
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Total number of triples: 438.