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filingDate 2003-07-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2005-12-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2005536494-A
titleOfInvention Substituted heterocycloderivatives and methods useful as antidiabetic and antiobesity agents
abstract [Formula 1] [Wherein Z 1 is (CH 2 ) q or C═O; Z 2 is (CH 2 ) p or C═O; D is —CH═, C═O or (CH 2 ) m and m is 0, 1, 2 or 3; n is 0, 1 or 2; p is 1 or 2; q is 0, 1 or 2; Q is C or N; A is (CH 2 ) x and x is 1 to 5, or A Is (CH 2 ) x 1 and x 1 is 1 to 5 and may contain an alkenyl or alkynyl bond anywhere in the chain; or A is — (CH 2 ) x 2 —O— (CH 2 ) x 3 -and x 2 is 0 to 5, and x 3 is also 0 to 5, but at least one of x 2 and x 3 is not 0; B is a bond or (CH 2 ) x 4 x 4 is 1 to 5; X is CH or N; X 2 is C, N, O or S; X 3 is C, N, O or S; X 4 is C, N, O or S; X 5 Is C, N, O or S; X 6 is C, N, O or S; provided that at least one of X 2 , X 3 , X 4 , X 5 and X 6 is N; and X 2 , X 3, X 4, out of X 5 and X 6 One even without is C. R 1 is H or alkyl; R 2 is H, alkyl, alkoxy, halogen, amino, substituted amino or cyano; R 2a , R 2b and R 2c are the same or different and H, alkyl, alkoxy, halogen, amino, substituted amino Or cyano; R 3 , E, Z and Y are as defined in the specification. ] The compound of.
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Total number of triples: 1388.