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filingDate 2003-01-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2005-07-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2005521674-A
titleOfInvention Manufacture of oral dosage forms that deliver immediate and sustained release drugs
abstract Disclosed is a method for producing a pharmaceutical tablet for oral administration, wherein the tablet combines both immediate and sustained mode drug delivery and is an immediate drug that is insoluble or only slightly soluble in water And the immediate-acting drug is present in very small amounts compared to the long-acting drug. The method includes the use of immediate-acting drug particles having a diameter of 10 μm or less applied as a layer or coating on a long-acting drug core, wherein the layer or coating is an aqueous suspension or Or any drug particle itself applied as a solid mixture containing the drug as a mixture with a material that disintegrates rapidly in gastric juice. In any case, the results have a high degree of uniformity in the ratio of immediate drug and long-acting drug, taking into account the insolubility of the fast-acting drug and the relatively small amount of immediate-acting drug compared to the long-acting drug, Uniformity is difficult to achieve otherwise.
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