http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2481726-A2

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publicationDate 2012-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-2481726-A2
titleOfInvention Crystal forms of saxagliptin and processes for preparing same
abstract Physical crystal structures of a compound of the formula (I): are provided including the free base monohydrate thereof (form H-1) and the hydrochloric acid salt thereof, including hydrochloric acid salt containing 0.75 equivalent of H 2 O (form H0.75-3) and hydrochloric acid salt containing 2 equivalents of H 2 O (form H2-1), and hydrochloric acid salt Pattern P-5, preferably in substantially pure form, and other forms as described herein, pharmaceutical compositions containing structures of compound I or IA, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures.
priorityDate 2007-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1201.