Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_dfd617dc43a4c986d2dd81e4cb39d9dd |
classificationCPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B2200-07 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-09 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-16 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B53-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-09 |
filingDate |
2004-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9308340b52d13991a456d71863132429 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4962d02ab4fef1f4000ee7288bb079d5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_93e25445ad46a6a91947090b6c3ddff2 |
publicationDate |
2008-06-18-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
EP-1693364-A4 |
titleOfInvention |
INTERMEDIATES FOR THE PRODUCTION OF OPTICALLY ACTIVE CYCLOPROPYLAMINE DERIVATIVES AND PROCESS FOR THE PRODUCTION THEREOF |
abstract |
Provided are a process for the production of intermediates from which optically active cyclopropylamine derivatives (6) can be easily synthesized by a short operation without optical resolution; and such intermediates. A process for the production of optically active compounds represented by the general formula (4) or salts thereof: (4) (wherein R1 is an amino-protecting group), characterized by reacting an optically active compound represented by the general formula (3): (3) (wherein R1 is as defined above) with a reagent prepared from both a titanium(IV) reagent and an alkylmetal compound, if necessary, in the presence of a Lewis acid. |
priorityDate |
2003-12-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |