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filingDate 1990-07-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1992-01-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber EP-0468121-A1
titleOfInvention Process for the galenical preparation of a therapeutic composition, in particular based on aspirin
abstract - de mise en solution du principe actif de départ dans un solvant approprié, - d'imprégnation de la solution ainsi formée sur un support alimentaire de structure appropriée et pharmaceutiquement compatible avec ledit principe actif, - d'évaporation du solvant de la solution adsorbée au sein dudit support en provoquant la reconstitution du principe actif par la formation de microcristaux adsorbés sur les parois et au sein du substrat, - et le procédé est caractérisé en ce que le solvant est constitué d'un système binaire comportant un solvant principal, de nature organique, et un adjuvant, de type solide à la température ambiante et soluble dans le solvant principal, l'adjuvant présentant par ailleurs des propriétés lubrifiantes Process for the preparation of a therapeutic composition for internal use, in particular for administration per os, in galenical presentation, and containing at least one active principle in solid form adsorbed on a substrate, the active product being distributed therein in the form of microparticles finely dispersed and the process being of the type comprising the phases: - dissolving the starting active principle in an appropriate solvent, - impregnating the solution thus formed on a food support of appropriate structure and pharmaceutically compatible with said active ingredient, - evaporation of the solvent from the solution adsorbed within said support, causing the active principle to be reconstituted by the formation of microcrystals adsorbed on the walls and within the substrate, - And the process is characterized in that the solvent consists of a binary system comprising a main solvent, of organic nature, and an adjuvant, of solid type at room temperature and soluble in the main solvent, the adjuvant having by elsewhere lubricating properties
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