Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_3cadfb09acd5bddac739df8e712442b0 |
classificationCPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K45-06 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K45-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-437 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-437 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-46 |
filingDate |
2016-12-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_45304ccaa92e65a668b136c0415f6a08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3e5315a76207fd3878c98be95b005dc6 |
publicationDate |
2018-09-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
CN-108602821-A |
titleOfInvention |
1H-imidazo[4,5-B]pyridyl and 2-oxo-2,3-dihydro-1H-imidazo[4,5-B]pyridyl heterocyclic BET bromodomain inhibitors |
abstract |
Disclosed herein are substituted 1H-imidazo[4,5-b]pyridyl and 2-oxo-2,3-dihydro-1H-imidazolo which are useful as inhibitors of BET protein function by binding to bromodomains [4,5-b]pyridyl heterocyclic compounds, compositions comprising said compounds and their use in therapy. These compounds are useful in the treatment of diseases and conditions such as cancer, autoimmune disease, inflammation and cardiovascular disease. |
isCitedBy |
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-113264930-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-113264930-B |
priorityDate |
2015-12-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |