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filingDate 2010-05-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b7d3ac2c5f0ab7e111d798c51d4ce0d9
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publicationDate 2014-07-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber CN-103896796-A
titleOfInvention Substituted aminopropionic acid derivatives as neprilysin inhibitors
abstract A substituted alanine derivative as a neprilysin inhibitor. The present invention provides a compound of formula I', or a pharmaceutically acceptable salt thereof, wherein R 1 , R 2 , R 3 , R 5 , B 1 , X and n are as defined herein. The invention also relates to processes for the preparation of the compounds of the invention and their therapeutic use. The present invention further provides a combination of pharmacologically active agents and a pharmaceutical composition.
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priorityDate 2009-05-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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