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Woltering TJ, Wichmann J, Goetschi E, Adam G, Kew JNC, Knoflach F, Ballard TM, Huwyler J, Mutel V, Gatti S. Synthesis and characterization of 1,3-dihydro-benzo[b][1,4]diazepin-2-one derivatives: Part 3. New potent non-competitive metabotropic glutamate receptor 2/3 antagonists. Bioorganic & Medicinal Chemistry Letters. 2008 Apr;18(8):2725–9. doi: 10.1016/j.bmcl.2008.02.076. |