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Pignatello R, Guccione S, Forte S, Di Giacomo C, Sorrenti V, Vicari L, Uccello Barretta G, Balzano F, Puglisi G. Lipophilic conjugates of methotrexate with short-chain alkylamino acids as DHFR inhibitors. Synthesis, biological evaluation, and molecular modeling. Bioorg Med Chem. 2004 Jun 01;12(11):2951–64. doi: 10.1016/j.bmc.2004.03.040. PMID: 15142554. |