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Ballet S, Feytens D, Wachter RD, Vlaeminck MD, Marczak ED, Salvadori S, Graaf CD, Rognan D, Negri L, Lattanzi R, Lazarus LH, Tourwé D, Balboni G. Conformationally constrained opioid ligands: The Dmt-Aba and Dmt-Aia versus Dmt-Tic scaffold. Bioorganic & Medicinal Chemistry Letters. 2009 Jan;19(2):433–7. doi: 10.1016/j.bmcl.2008.11.051. |