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Fish PV, Barta NS, Gray DLF, Ryckmans T, Stobie A, Wakenhut F, Whitlock GA. Derivatives of (3S)-N-(biphenyl-2-ylmethyl)pyrrolidin-3-amine as selective noradrenaline reuptake inhibitors: Reducing P-gp mediated efflux by modulation of H-bond acceptor capacity. Bioorganic & Medicinal Chemistry Letters. 2008 Aug;18(15):4355–9. doi: 10.1016/j.bmcl.2008.06.071. |