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Pascal Y, Andrianjara CR, Auclair E, Avenel N, Bertin B, Calvet A, Féru F, Lardon S, Moodley I, Ouagued M, Payne A, Pruniaux M, Szilagyi C. Synthesis and structure–activity relationships of 4-oxo-1-phenyl-3,4,6,7-tetrahydro-[1,4]diazepino[6,7,1- hi ]indoles: novel PDE4 inhibitors. Bioorganic & Medicinal Chemistry Letters. 2000 Jan;10(1):35–8. doi: 10.1016/s0960-894x(99)00573-9. |