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Jeffries B, Wang Z, Felstead HR, Le Questel JY, Scott JS, Chiarparin E, Graton J, Linclau B. Systematic Investigation of Lipophilicity Modulation by Aliphatic Fluorination Motifs. J Med Chem. 2020 Feb 13;63(3):1002–31. doi: 10.1021/acs.jmedchem.9b01172. PMID: 31894985. |