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Mulvihill MJ, Ji Q, Werner D, Beck P, Cesario C, Cooke A, Cox M, Crew A, Dong H, Feng L, Foreman KW, Mak G, Nigro A, O’Connor M, Saroglou L, Stolz KM, Sujka I, Volk B, Weng Q, Wilkes R. 1,3-Disubstituted-imidazo[1,5-a]pyrazines as insulin-like growth-factor-I receptor (IGF-IR) inhibitors. Bioorganic & Medicinal Chemistry Letters. 2007 Feb;17(4):1091–7. doi: 10.1016/j.bmcl.2006.11.016. |