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Gandhi DM, Majewski MW, Rosas R, Kentala K, Foster TJ, Greve E, Dockendorff C. Characterization of Protease-Activated Receptor (PAR) ligands: Parmodulins are reversible allosteric inhibitors of PAR1-driven calcium mobilization in endothelial cells. Bioorganic & Medicinal Chemistry. 2018 May;26(9):2514–29. doi: 10.1016/j.bmc.2018.04.016. |