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Methot JL, Fischer C, Li C, Rivkin A, Ahearn SP, Brown WC, Kattar S, Kelley E, Mampreian DM, Schell A, Rosenau A, Zhou H, Ball R, Deshmukh SV, Jeliazkova-Mecheva VV, Diaz D, Moy LY, Kenific CM, Moxham C, Shah S, Nuthall H, Szewczak AA, Hill A, Hughes B, Smotrov N, Munoz B, Miller TA, Shearman MS. Potent benzoazepinone γ-secretase modulators with improved bioavailability. Bioorganic & Medicinal Chemistry Letters. 2015 Sep;25(17):3495–500. doi: 10.1016/j.bmcl.2015.06.032. |