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Zhu R, Seow HA, Baumann RP, Ishiguro K, Penketh PG, Shyam K, Sartorelli AC. Design of a hypoxia-activated prodrug inhibitor of O6-alkylguanine-DNA alkyltransferase. Bioorganic & Medicinal Chemistry Letters. 2012 Oct;22(19):6242–7. doi: 10.1016/j.bmcl.2012.08.008. |