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Ding F, Shen HC, Wilsie LC, Krsmanovic ML, Taggart AK, Ren N, Cai T, Wang J, Tong X, Holt TG, Chen Q, Gerard Waters M, Hammond ML, Tata JR, Colletti SL. Discovery of pyrazolyl propionyl cyclohexenamide derivatives as full agonists for the high affinity niacin receptor GPR109A. Bioorganic & Medicinal Chemistry Letters. 2010 Jun;20(11):3372–5. doi: 10.1016/j.bmcl.2010.04.013. |