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Colabufo NA, Abate C, Contino M, Inglese C, Ferorelli S, Berardi F, Perrone R. Tritium radiolabelling of PB28, a potent sigma-2 receptor ligand: pharmacokinetic and pharmacodynamic characterization. Bioorganic & Medicinal Chemistry Letters. 2008 Mar;18(6):2183–7. doi: 10.1016/j.bmcl.2007.12.056. |