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Woltering TJ, Adam G, Wichmann J, Goetschi E, Kew JNC, Knoflach F, Mutel V, Gatti S. Synthesis and characterization of 8-ethynyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one derivatives: Part 2. New potent non-competitive metabotropic glutamate receptor 2/3 antagonists. Bioorganic & Medicinal Chemistry Letters. 2008 Feb;18(3):1091–5. doi: 10.1016/j.bmcl.2007.12.005. |