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Chenard BL, Lipinski CA, Dominy BW, Mena EE, Ronau RT, Butterfield GC, Marinovic LC, Pagnozzi M, Butler TW, Tsang T. A unified approach to systematic isosteric substitution for acidic groups and application to NMDA antagonists related to 2-amino-7-phosphonoheptanoate. J Med Chem. 1990 Mar;33(3):1077–83. doi: 10.1021/jm00165a030. PMID: 2155321. |