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Chen H, Boiziau J, Parker F, Mailliet P, Commerçon A, Tocque B, Le Pecq JB, Roques BP, Garbay C. Structure-activity relationships in a series of 5-[(2,5-dihydroxybenzyl)amino]salicylate inhibitors of EGF-receptor-associated tyrosine kinase: importance of additional hydrophobic aromatic interactions. J Med Chem. 1994 Mar 18;37(6):845–59. doi: 10.1021/jm00032a020. PMID: 8145236. |