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Koolpe GA, Nelson WL, Gioannini TL, Angel L, Appelmans N, Simon EJ. Opioid agonists and antagonists. 6-Desoxy-6-substituted lactone, epoxide, and glycidate ester derivatives of naltrexone and oxymorphone. J Med Chem. 1985 Jul;28(7):949–57. doi: 10.1021/jm00145a018. PMID: 2409280. |