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Briguglio I, Laurini E, Pirisi MA, Piras S, Corona P, Fermeglia M, Pricl S, Carta A. Triazolopyridinyl-acrylonitrile derivatives as antimicrotubule agents: Synthesis, in vitro and in silico characterization of antiproliferative activity, inhibition of tubulin polymerization and binding thermodynamics. European Journal of Medicinal Chemistry. 2017 Dec;141():460–72. doi: 10.1016/j.ejmech.2017.09.065. |