bibliographicCitation |
Gonzalez-Lopez de Turiso F, Hao X, Shin Y, Bui M, Campuzano IDG, Cardozo M, Dunn MC, Duquette J, Fisher B, Foti RS, Henne K, He X, Hu Y, Kelly RC, Johnson MG, Lucas BS, McCarter J, McGee LR, Medina JC, Metz D, San Miguel T, Mohn D, Tran T, Vissinga C, Wannberg S, Whittington DA, Whoriskey J, Yu G, Zalameda L, Zhang X, Cushing TD. Discovery and in Vivo Evaluation of the Potent and Selective PI3Kδ Inhibitors 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-6-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-0687) and 2-((1S)-1-((6-Amino-5-cyano-4-pyrimidinyl)amino)ethyl)-5-fluoro-N-methyl-3-(2-pyridinyl)-4-quinolinecarboxamide (AM-1430). J. Med. Chem. 2016 Jul 25;59(15):7252–67. doi: 10.1021/acs.jmedchem.6b00827. |