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Hasegawa F, Kawamura K, Tsuchikawa H, Murata M. Stable C-N axial chirality in 1-aryluracil scaffold and differences in in vitro metabolic clearance between atropisomers of PDE4 inhibitor. Bioorg Med Chem. 2017 Aug 15;25(16):4506–11. doi: 10.1016/j.bmc.2017.06.042. PMID: 28698053. |