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Tanaka M, Chiba K, Okita M, Kaneko T, Tagami K, Hibi S, Okamoto Y, Shirota H, Goto M, Sakurai H. 3-(5-Alkyl-4-hydroxy-3-methoxy-1-naphthalenyl)-2-methyl-2-propenoic acids as orally active inhibitors of IL-1 generation. J Med Chem. 1991 Aug;34(8):2647–9. doi: 10.1021/jm00112a046. PMID: 1875355. |