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Hay DL, Christopoulos G, Christopoulos A, Sexton PM. Determinants of 1-Piperidinecarboxamide,N-[2-[[5-Amino-l-[[4-(4-pyridinyl)-l-piperazinyl]carbonyl]pentyl]amino]-1-[(3,5-dibromo-4-hydroxyphenyl)methyl]-2-oxoethyl]-4-(1,4-dihydro-2-oxo-3(2H)-quinazolinyl) (BIBN4096BS) Affinity for Calcitonin Gene-Related Peptide and Amylin Receptors—The Role of Receptor Activity Modifying Protein 1. Mol Pharmacol. 2006 Sep 07;70(6):1984–91. doi: 10.1124/mol.106.027953. |