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Nishizawa R, Nishiyama T, Hisaichi K, Minamoto C, Matsunaga N, Takaoka Y, Nakai H, Jenkinson S, Kazmierski WM, Tada H, Sagawa K, Shibayama S, Fukushima D, Maeda K, Mitsuya H. Spirodiketopiperazine-based CCR5 antagonist: Discovery of an antiretroviral drug candidate. Bioorganic & Medicinal Chemistry Letters. 2011 Feb;21(4):1141–5. doi: 10.1016/j.bmcl.2010.12.109. |