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filingDate 1995-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_06621caa512de897df69b4312636679b
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publicationDate 1996-04-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-9609820-A1
titleOfInvention Inhibitors of farnesyl-protein transferase
abstract The present invention comprises dipeptide analogs that inhibit the farnesylation of Ras. These farnesyl-protein transferase inhibitors are characterized by the inclusion of a cyclic amine in the backbone of the dipeptide. Further contained in this invention are chemotherapeutic compositions containing these farnesyl transferase inhibitors and methods for their production.
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Total number of triples: 445.