http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-9602239-A2

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filingDate 1995-07-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1996-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-9602239-A2
titleOfInvention Enhanced loading of solutes into polymer gels and methods of use
abstract A method of loading a drug into a crosslinked polymer network and protecting the drug from the effects of inactivation is described. The method includes the steps of contacting of a biologically active solute (i.e., drug) with: (i) a gel network; (ii) a second protectant polymer that is somewhat immiscible with the gel; and (iii) a protectant salt, under conditions sufficient for the biologically active solute to selectively partition into the gel and the protectants to be entrained in the gel. A drug delivery system is also described. It comprises a polymer gel network including the drug to be delivered; protectants including a salt and a loading polymer, the salt and the loading polymer capable of protecting the drug from loss of activity. The polymer gel network is capable of expanding or collapsing in response to a change in an environmental condition to which the gel is exposed, the expanding or collapsing sufficient to release the drug into an environment of use.
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Total number of triples: 1827.