http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-9302674-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_07b71571160c289fbf5fc680dfea513f |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D233-64 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F7-1804 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C271-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C271-18 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F7-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C271-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C271-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D233-54 |
| filingDate | 1992-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a213f4e54a97f55560b9a62e55e6b7ad http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ffbe8099b8ac45b38084c58934e5848a |
| publicationDate | 1993-02-18-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | WO-9302674-A1 |
| titleOfInvention | Hiv protease inhibitors |
| abstract | Compounds of formula (I), wherein R?1, R1', R3, R4, R5¿ are independently H, C¿1-6?alkyl, C2-6alkenyl, C3-7cycloalkyl, Ar, Het, T-C1-6alkyl, T-C2-6alkenyl; T is Ar, Het or C3-7cycloalkyl; R?2¿ is Y, (CHR4)n-Y, =CR5(CHR4)n-Y; R3 is H, OH; Q is OH or NH¿2?; W is R?6, R6CO, R6OCO, R6OCH(R7)CO, R6NHCH(R7)CO, R6SCH(R7)CO, R6SO¿2, R6SO or an amino acid with a blocked or unblocked amino terminus; R?6 and R7¿ are independently H, C¿1-6?alkyl, C3-7cycloalkyl, Ar, Het, T-C1-6alkyl, T-(CH2)nCH(T)(CH2)n; X is (H,OH) or =O; Y is H; OH, NR'R?4¿, Ar, Het or CO-Z; Z is OH, NR'R4, OR4 or an amino acid with a blocked or unblocked carboxy terminus; R' is H, C¿1-6?alkyl, Ar-C1-6alkyl; n is 1 to 4; and pharmaceutically acceptable salts thereof, are inhibitors of the HIV-1 protease and are useful in the treatment of AIDS. |
| isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-7115652-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-7132568-B2 |
| priorityDate | 1991-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 254.