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filingDate 1992-03-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1992-10-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-9216226-A1
titleOfInvention Il-1 inhibitors
abstract The present invention provides for a novel mechanism of controlling anti-inflammatory activity in a mammal, including humans. The inhibition of P-glycoprotein mediated transport of Interleukin-1 (IL-1) from cells, by an inhibitor of the mdr P-glycoprotein, provides for treatment of indications in which excessive extracellular IL-1 activity is implicated. Such activity has been implicated in such disease as rheumatoid arthritis and osteoarthritis.
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