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filingDate 1990-03-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6a631b4a32ae9e43380e3601220e9ef8
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_13b2d728247130657135e03f717a324d
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6ba0026b6933dcceeaa41f36b2c7283b
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_648546a4ab523ae0bfdeef314657f053
publicationDate 1990-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-9010649-A1
titleOfInvention Serpin resistant chymotrypsin superfamily proteases, particularly pai-1 resistant +-pa, complementary inhibitor mutants; compositions; genes; expression
abstract The present invention relates to serine protease mutants of the chymotrypsin superfamily, particularly +-PA mutants, that are resistant to inhibition by their cognate inhibitors, such as PAI-1 in the case of +-PA, and genes that encode the same. The present invention also relates to serine protease inhibitor mutants, particularly PAI-1 mutants, that inhibit the serine protease mutants of the present invention, particularly +-PA mutants, and genes that encode the same. The serine protease mutants and serine protease inhibitor mutants are useful as, e.g., pharmacological agents.
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Total number of triples: 566.