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filingDate 1988-08-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 1989-03-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-8901779-A1
titleOfInvention Molecular decoyants and methods of use thereof
abstract Molecular decoyants are chemical structures which functionally resemble an endogenous receptor. They may be used for the treatment of humans or other animals which have been subjected to a foreign agent which exerts an undesired effect only after first binding to that endogenous receptor. A decoyant is a fraction of an endogenous receptor which retains the essential elements of the binding site of the receptor for the foreign agent or is a synthetic or biosynthetic derivative thereof. The alpha-184-200 amino acid sequence of Torpedo californica acetylcholine receptor is an example of a decoyant which protects against curarimimetic neurotoxins. Another example is the fraction of the CD4 receptor which retains the essential elements of the receptor for protection against HIV.
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