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filingDate 2022-04-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8d75fc8ab07d8672e737bb4a02a9a805
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5c3a6a6dae1e8cba3b0ee7497e57bc2e
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publicationDate 2022-12-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2022255915-A1
titleOfInvention Pet radiotracers
abstract The compounds of the invention are ASEM analogs with different ortho- and para-substitutions that can be labelled with 3H and/or 11C to be used as PET radiotracers capable of binding to α7-nAChR both in vitro and in vivo in a subject body. The PET radiotracers thereby enable visualization and quantification of α7-nAChR in various target tissues, including monitoring the distribution of α7-nAChRs in such a target tissue. The compounds exhibit of high binding affinity and specificity towards α7-nAChR and are able to pass the blood-brain barrier (BBB).
priorityDate 2021-06-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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