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filingDate 2022-05-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_aa28f9c4e756ec85aad782a2b964d644
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publicationDate 2022-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2022236136-A1
titleOfInvention Exatecan derivatives and antibody-drug conjugates thereof
abstract Disclosed herein, in part, are compounds (I) which are exatecan derivatives with novel chemical linkers that include cathepsin B cleavable moieties, and conjugated to targeting antibodies.
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