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publicationDate 2022-09-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2022192745-A1
titleOfInvention Mta-cooperative prmt5 inhibitors
abstract Disclosed are compounds of Formula IIA, IIA-1, IIB, IIB-1, IIC and IIC-1: and pharmaceutical compositions and methods of use thereof These compounds inhibit Protein Arginine M-Methyl Transferase 5 (PRMT5) activity and are useful in methods and pharmaceutical compositions for treating cancer.
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Total number of triples: 1129.