http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2022166993-A1

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-69
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
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filingDate 2022-02-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_34e40b0908d0f2cf713372ab86bf4ca8
publicationDate 2022-08-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2022166993-A1
titleOfInvention Novel boron carrier, preparation method and pharmaceutical formulation thereof
abstract Disclosed in the present invention are a novel boron carrier, a preparation method and a pharmaceutical formulation thereof; in particular, the present invention relates to 3,4-dihydro-3-methyl-4-oxoimidazo[5,1-D]-1,2,3,5-tetrazine-8-carboxylic acid [4-(4,4,5,5-tetramethyl-1,3,2-diazaborolan-2-yl)phenyl ester, a preparation method and a pharmaceutical formulation thereof. The boron carrier compound (I) of the present invention has the advantages of stable quality, has excellent activity compared with the same type of medicines, is suitable for being developed as a novel boron carrier, and is suitable for preparing various forms of pharmaceutical formulations. Therefore, the boron carrier of the present invention has a good application prospect in preparation of medicines for treating tumors.
priorityDate 2021-02-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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