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filingDate 2021-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9581e4d227a450f61ead933bd1363a32
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publicationDate 2022-06-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2022123009-A1
titleOfInvention Method for manufacturing an inhalable powder comprising voriconazole
abstract The present invention relates to a method for manufacturing an inhalable powder comprising leucine and voriconazole or a pharmaceutically active salt thereof, in substantially crystalline form, in an amount greater than 50% by weight with respect to the total weight of the powder. The method comprises a first step consisting of providing a solution of voriconazole or pharmaceutically active salt thereof and leucine in a suitable vehicle, a second step consisting in drying said powder using the spray drying technique at an outlet temperature from 40 and 75°C and at a feed rate greater than 10 g/minute and finally collecting the powder obtained.
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