Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_bcb146c68b67089013b4c7a614504254 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_3e035457406455ea05989c01cb90c8f1 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D519-00 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P37-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D519-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4162 |
filingDate |
2021-10-19-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a5e6990bcc74a6210f798537fa7ce0c9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_65439aa70b41bfd70a861fff1f654ceb http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0d80141a40912e0dda33a8d75dfccc91 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eed3c5a9bd11136058195947309692aa http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_836c13d8cc9ab5fec8d89e49d635cc5f http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b6a9b069a5927e0316b28c1337b398e0 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_175ddae8ea20a4e957ea438ba4342690 |
publicationDate |
2022-05-19-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
WO-2022101603-A1 |
titleOfInvention |
Improved small molecules |
abstract |
This invention particularly relates to trifunctional PROTACs of formula I as described herein which bind to a protein within the Bromo- and Extra-Terminal (BET) family of proteins, and especially to PROTACs including small molecule E3 ubiquitin ligase protein binding ligand compounds which induce preferential degradation of the BRD2 protein within the bromodomain of the BET family of proteins. |
isCitedBy |
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-111741769-A |
priorityDate |
2020-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |