http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2022096679-A1

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filingDate 2021-11-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f49d663be9e427524002211707aff195
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b664f439fd689a0f5be2576b6ea5e9ce
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publicationDate 2022-05-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2022096679-A1
titleOfInvention Protein-protein interaction modulators of aurora kinase a and their use in the prevention and/or treatment of cancer
abstract The present invention relates to compounds that modulate the conformation of Aurora Kinase A (AURKA). The compounds of the present invention are also modulators of the interactome of AURKA, and preferably alter the protein-protein interaction of AURKA with binding proteins, such as MYC and/or TPX2. The present invention also pertains to the use of such compounds in the prevention and/or treatment of proliferative diseases, such as cancer, and kits comprising the same.
priorityDate 2020-11-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID294739
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID30590
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2331
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5365800

Total number of triples: 318.