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publicationDate 2022-03-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2022056281-A1
titleOfInvention Protein tyrosine phosphatase inhibitors and methods of use thereof
abstract Provided herein are compounds including compounds of formula (I), compositions, and methods useful for inhibiting protein tyrosine phosphatase, e.g., protein tyrosine phosphatase non-receptor type 2 (PTPN2) and/or protein tyrosine phosphatase non-receptor type 1 (PTPN1), and for treating related diseases, disorders and conditions favorably responsive to PTPN1 or PTPN2 inhibitor treatment,e.g., a cancer or a metabolic disease.
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