http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2021089845-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_b9ca0632596f3342a71f604d9152b9e1
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-166
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-5415
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-5415
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-166
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-02
filingDate 2020-11-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4814a44e384036fa111ad5a931159924
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5480b1968fb1c0873f72de8caeb4e075
publicationDate 2021-05-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2021089845-A1
titleOfInvention Cd93 inhibitors for use in the treatment of cancer
abstract The present invention relates to compounds of formula (1): Ar-L-N(R1)(R2), for use in the treatment of cancer. The compounds of formula (1) are characterized by a mono-, bi- or tricyclic aryl or heteroaryl (Ar) and a basic nitrogen atom with R1 and R2 being a linear alkyl or forming an aliphatic or heterocyclic ring. The aryl or heteroaryl and the basic nitrogen atom are connected via a linker L. The compounds of formula (1) are potent inhibitors of CD93, particularly of the CD93 intracellular domain.
priorityDate 2019-11-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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