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filingDate 2020-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2859a2f605dbe30ffe1c05556be1ef32
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publicationDate 2021-04-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2021059220-A1
titleOfInvention Process for the production of 5-(4-((2 s,5 s)-5-(4-chlorobenzyl)-2-methylmorpholino)piperidin-1-yl)-1 h-1,2,4-triazol-3-amine
abstract The present invention relates to a process for the synthesis of 5-(4-((2S,5S)-5-(4-chlorobenzyl)- 2-methylmorpholino)piperidin-1-yl)-1 H -1,2,4-triazol-3-amine in two hydrated crystalline forms and in one anhydrous crystalline form. The present invention further relates to methyl (Z)-4-((2S,5S)-5-(4-chlorobenzyl)-2-methylmorpholino)- N -cyanopiperidine-1-carbimidothio-ate which is an intermediate in this process.
priorityDate 2019-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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