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filingDate 2020-09-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e5bda28c08f8d1c134207e623852f999
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_48df2be6e4b2556728658186688563c7
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publicationDate 2021-04-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2021058017-A1
titleOfInvention Degradation of androgen receptor (ar) by conjugation of ar antagonists with e3 ligase ligand and methods of use
abstract Provided herein are novel bifunctional compounds formed by conjugating AR antagonist moieties with E3 ligase Ligand moieties, which function to recruit targeted proteins to E3 Ubiquitin ligase for degradation, and methods of preparation and uses thereof.
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Total number of triples: 1416.