http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2020243777-A1

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filingDate 2020-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3ee13f7f28c3438f9f786a7116ea0f5d
publicationDate 2020-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2020243777-A1
titleOfInvention Pharmaceutical formulations and systems for delivery of an androgenic agent and an aromatase inhibitor and methods for use
abstract The present disclosure is directed formulations, delivery systems and/or methods of use that have a novel a sustained release multi-phasic concentration pattern that may be used, among other things, for reducing mammographic breast density and/or breast stiffness in warm-blooded animals. For example, the formulation may comprise: the administration of an effective amount of androgenic agent and an effective amount of an aromatase inhibitor to a subject that provides a sustained release multi-phasic concentration pattern in the blood of the subject over time as measured by serum concentration for the androgen and plasma concentration for the aromatase inhibitor and improves, amoung other things, breast tissue stabilization and/or increases of the levels of androgen receptor expression. The present disclosure is also directed to the use of an effective amount of an androgenic agent in combination with an effective amount of an aromatase inhibitor for the prophylaxis or treatment of autoimmune inflammatory mastitis (AIM) in a patient in 15 need thereof. Autoimmune inflammatory mastitis includes the conditions of idiopathic inflammatory macromastia, plasma cell mastitis, granulomatous mastitis.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP96084
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Z1N4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP56560
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3902
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP18109
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21396
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ69FB6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI4
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID9606
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394204
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11048
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395097
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6YI21
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6YK33
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07453
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396580
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100009712
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24775
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID542014
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394205
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID23827
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJT9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15324
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07492
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJU0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID50943
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID398459
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCNP_112503
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6462
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22443
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395836
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68243
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9W7R2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5430
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8094
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68245
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04278
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20415
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8BW75
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395835
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID728378
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4784
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF6QRS1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A1L9WUM2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID450133

Total number of triples: 357.