http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2020168170-A1

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filingDate 2020-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_78cd885fe95adcae094fdaca8897fabe
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a32c23c54acf0ed557a8d13f3ea6bbb9
publicationDate 2020-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2020168170-A1
titleOfInvention Isotopically-stabilized tetronimide compounds
abstract Isotopically-stabilized tetronimide compounds comprising one or more deuterium atoms, derivatives, and intermediates, thereof, including methods for their synthesis, pharmaceutical compositions thereof, and methods of using these compounds to interact with target molecules in cell-free samples, cell- and tissue-based assays, animal models, and in a subject are disclosed. One aspect relates to molecules that modulate the expression or catalytic activity of aspartyl (asparaginyl) β-hydroxylase (ASPH) within or on the surface of a cell. Other aspects of the invention relate to use of the molecules disclosed herein to diagnose, ameliorate, or treat cell proliferation disorders and related diseases. Related aspects include uses of the compounds to modulate the activity of viruses, as anti¬ hyperlipidemia agents, and as agents to ameliorate or treat thrombosis and related cardiovascular and metabolic disorders.
priorityDate 2019-02-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457781088
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22178470
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID476104
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25268
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID73506471
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID461435
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6251
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1PI70
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Total number of triples: 839.