http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2020166820-A1

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filingDate 2020-01-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_367b7ecf53d47c43692df4c225f79968
publicationDate 2020-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2020166820-A1
titleOfInvention Composition for subcutaneous injection containing microparticles comprising finasteride
abstract The present invention provides a composition for subcutaneous injection containing microparticles comprising finasteride, the composition comprising: microparticles comprising finasteride and biodegradable polymer; and a suspension solvent. The composition for subcutaneous injection of the present invention is provided in a subcutaneously injectable form, not in an oral administration form, and thus there is no need for a user to store the composition, and a hair loss treatment effect by finasteride can be exhibited through a method of direct administration at a hospital, and thus ease of storage and handling is excellent. When microparticles comprising finasteride are administered using the composition for subcutaneous injection of the present invention, a long-term drug administration effect over a period of 1-3 months can be maintained. In addition, in the present invention, as the diameter of particles is formed to a uniform micro-size, the release of a drug from microparticles is controlled, thereby enabling an effective drug concentration to be constantly maintained, and the present invention can be provided as a composition for injection, in which, when applied to an injection consisting of a uniform size of particles and administered as an injection to a patient, the sense of foreign matter and pain are reduced.
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